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A selenide linker for "traceless" solid-phase organic synthesis

A selenide linker for "traceless" solid-phase organic synthesis
A selenide linker for "traceless" solid-phase organic synthesis
4-Bromophenethyl alcohol was protected as the THP ether, followed by reaction with magnesium and selenium to give the corresponding diselenide. Ether deprotection provides a diselenide diol, which is attached to solid-phase resins. The polymer-bound selenide anion is then generated, and functions as a traceless linker for electrophiles such as alkyl halides.
solid-phase synthesis, traceless linkers, selenides strategies, cleavage
0006-3592
104-106
Li, Z. G.
166e9d42-b238-4112-8145-8172a3d024ea
Kulkarni, B. A.
780354e8-3ad9-49fa-96a5-8f5890179306
Ganesan, A.
62aa5a87-9308-4383-8686-99726b6bcfb9
Li, Z. G.
166e9d42-b238-4112-8145-8172a3d024ea
Kulkarni, B. A.
780354e8-3ad9-49fa-96a5-8f5890179306
Ganesan, A.
62aa5a87-9308-4383-8686-99726b6bcfb9

Li, Z. G., Kulkarni, B. A. and Ganesan, A. (2000) A selenide linker for "traceless" solid-phase organic synthesis. Biotechnology and Bioengineering, 71 (2), 104-106. (doi:10.1002/1097-0290(2000)71:2<104::AID-BIT1000>3.0.CO;2-7).

Record type: Article

Abstract

4-Bromophenethyl alcohol was protected as the THP ether, followed by reaction with magnesium and selenium to give the corresponding diselenide. Ether deprotection provides a diselenide diol, which is attached to solid-phase resins. The polymer-bound selenide anion is then generated, and functions as a traceless linker for electrophiles such as alkyl halides.

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More information

Published date: 2000
Keywords: solid-phase synthesis, traceless linkers, selenides strategies, cleavage

Identifiers

Local EPrints ID: 18917
URI: http://eprints.soton.ac.uk/id/eprint/18917
ISSN: 0006-3592
PURE UUID: e68a84dc-2ab0-412f-913c-e251f6546c4a

Catalogue record

Date deposited: 18 Jan 2006
Last modified: 15 Mar 2024 06:09

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Contributors

Author: Z. G. Li
Author: B. A. Kulkarni
Author: A. Ganesan

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