Bevacqua, F., Basso, A., Gitto, R., Bradley, M. and Chimirri, A.
Solid-phase Friedel-Crafts acylation on polystyrene resins-synthesis of antiepiletic 1-aryl-3,5-dihydro-4H-2,3-benzodiazepin-4-ones
Tetrahedron Letters, 42, (43), . (doi:10.1016/S0040-4039(01)01602-1).
Full text not available from this repository.
Friedel-Crafts acylation with various acyl chlorides of resin-bound 3,4-dimethoxyphenylacetate afforded resin bound ketones which, following treatment with hydrazine, were converted into the corresponding 2,3-benzodiazepines in good yields and purities.
Actions (login required)