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A bifunctional antibody targeting PD-1 and TGF-β signaling has antitumor activity in combination with radiotherapy and attenuates radiation-induced lung injury

A bifunctional antibody targeting PD-1 and TGF-β signaling has antitumor activity in combination with radiotherapy and attenuates radiation-induced lung injury
A bifunctional antibody targeting PD-1 and TGF-β signaling has antitumor activity in combination with radiotherapy and attenuates radiation-induced lung injury
Radio-immunotherapy has antitumor activity but also causes toxicity, which limits its clinical application. JS-201 is a dual antibody targeting PD-1 and TGF-β signaling. We investigated the antitumour effect of JS-201 combined with radiotherapy and the effect on radiation-induced lung injury (RILI). Different tumor models were established to detect the antitumor effects of the combination of JS-201 and RT, and RILI models were established to observe the effects of JS-201. Transcriptome sequencing showed that JS-201 optimized the TME by inhibiting extracellular matrix formation and angiogenesis. Combining JS-201 with radiotherapy further increased the inflammatory response and immune infiltration and showed great abscopal effects in LLC-luc models. Single-cell sequencing demonstrated that JS-201 reduced fibroblast proliferation by inhibiting the TGF-β/Smad pathway and the release of neutrophil extracellular traps mediated by ROS, thereby relieving radiation-induced pulmonary fibrosis. In conclusion, the JS-201 and radiotherapy combination enhances antitumor effects while mitigating acute and chronic RILI, and it may have potential for translational investigation as a cancer treatment strategy.
1158/2326-6066.CIR-23-0903
2326-6066
Wang, Sheng
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Xu, Duo
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Wang, Yuan
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Zhou, Yuehua
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Xiao, Lingyan
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Li, Fang
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Tu, Jingyao
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Qin, Wan
18ad2498-00e7-48fe-bcfa-b35355c66111
Tian, Sidan
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Zheng, Bolong
1d71f8fb-33e6-447b-94ce-784977948f76
Wang, Yihua
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Yuan, Xianglin
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Liu, Yuanhui
064a0c85-f930-4eac-b45c-7668477b8b13
Liu, Bo
e5628c10-c9d7-4fb7-ac7d-0334a0c75567
Wang, Sheng
cfcac135-9538-49d8-abfc-e452d3533a8f
Xu, Duo
47aa43bb-09d0-4aaa-9619-6a86e2d8afd1
Wang, Yuan
86f94a35-bd78-46d1-ab1b-4e1d3e033a59
Zhou, Yuehua
7d95e338-755a-4bf4-acbe-418720c3dedb
Xiao, Lingyan
1197ed66-06c8-4ad8-81cc-951239a32f5d
Li, Fang
5d22f265-dbda-4419-95c9-d2e1a84e9cd1
Tu, Jingyao
7cb601fb-6475-4dc0-8a83-f8d45e989bc1
Qin, Wan
18ad2498-00e7-48fe-bcfa-b35355c66111
Tian, Sidan
9c2df5a5-a4e5-4b20-aa83-99adfd8d981f
Zheng, Bolong
1d71f8fb-33e6-447b-94ce-784977948f76
Wang, Yihua
f5044a95-60a7-42d2-87d6-5f1f789e3a7e
Yuan, Xianglin
ec272d8a-ac62-4c0b-a835-9dda14169e01
Liu, Yuanhui
064a0c85-f930-4eac-b45c-7668477b8b13
Liu, Bo
e5628c10-c9d7-4fb7-ac7d-0334a0c75567

Wang, Sheng, Xu, Duo, Wang, Yuan, Zhou, Yuehua, Xiao, Lingyan, Li, Fang, Tu, Jingyao, Qin, Wan, Tian, Sidan, Zheng, Bolong, Wang, Yihua, Yuan, Xianglin, Liu, Yuanhui and Liu, Bo (2025) A bifunctional antibody targeting PD-1 and TGF-β signaling has antitumor activity in combination with radiotherapy and attenuates radiation-induced lung injury. Cancer Immunology Research, 2025. (1158/2326-6066.CIR-23-0903).

Record type: Article

Abstract

Radio-immunotherapy has antitumor activity but also causes toxicity, which limits its clinical application. JS-201 is a dual antibody targeting PD-1 and TGF-β signaling. We investigated the antitumour effect of JS-201 combined with radiotherapy and the effect on radiation-induced lung injury (RILI). Different tumor models were established to detect the antitumor effects of the combination of JS-201 and RT, and RILI models were established to observe the effects of JS-201. Transcriptome sequencing showed that JS-201 optimized the TME by inhibiting extracellular matrix formation and angiogenesis. Combining JS-201 with radiotherapy further increased the inflammatory response and immune infiltration and showed great abscopal effects in LLC-luc models. Single-cell sequencing demonstrated that JS-201 reduced fibroblast proliferation by inhibiting the TGF-β/Smad pathway and the release of neutrophil extracellular traps mediated by ROS, thereby relieving radiation-induced pulmonary fibrosis. In conclusion, the JS-201 and radiotherapy combination enhances antitumor effects while mitigating acute and chronic RILI, and it may have potential for translational investigation as a cancer treatment strategy.

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Accepted/In Press date: 24 January 2025
Published date: 29 January 2025

Identifiers

Local EPrints ID: 498507
URI: http://eprints.soton.ac.uk/id/eprint/498507
DOI: 1158/2326-6066.CIR-23-0903
ISSN: 2326-6066
PURE UUID: cd359777-0f04-4879-aa70-3e3ab998ccef
ORCID for Yihua Wang: ORCID iD orcid.org/0000-0001-5561-0648

Catalogue record

Date deposited: 20 Feb 2025 17:41
Last modified: 22 Aug 2025 02:13

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Contributors

Author: Sheng Wang
Author: Duo Xu
Author: Yuan Wang
Author: Yuehua Zhou
Author: Lingyan Xiao
Author: Fang Li
Author: Jingyao Tu
Author: Wan Qin
Author: Sidan Tian
Author: Bolong Zheng
Author: Yihua Wang ORCID iD
Author: Xianglin Yuan
Author: Yuanhui Liu
Author: Bo Liu

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