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A novel SPECT-CT imaging platform for quantifying in vivo lung cytokine signals in COPD

A novel SPECT-CT imaging platform for quantifying in vivo lung cytokine signals in COPD
A novel SPECT-CT imaging platform for quantifying in vivo lung cytokine signals in COPD
Introduction: disease-modifying treatments such as monoclonal antibodies can be highly effective in chronic inflammatory diseases such as COPD, but often fail in clinical trials due to heterogeneity of inflammation and imperfect tools to stratify patients to select optimal therapeutic approaches. Molecular imaging provides the potential to transform precision medicine in this field.

Methods: we developed and tested a novel molecular imaging platform using therapeutic monoclonal antibodies labelled with SPECT-CT detectable markers to quantify in vivo TNF involved in chronic lung inflammation in humans. We undertook a proof-of-concept clinical study involving participants with COPD and healthy controls. Participants underwent SPECT-CT imaging at 6- and 24-hours following injection of 99m-Tc-anti-TNF. Segmentation of lung regions and 99m-Tc-anti-TNF activity quantification was undertaken using novel semi-automated and AI-driven approaches.

Results: a significant increase in normalised activity, representing increased TNF inflammatory activity, was seen between the two time-points in the COPD group (64.88% +/- [SD] 31.04, p=.029) and not in healthy controls (35.38% +/- 34.33, =.110). However, analysis at a single time-point revealed higher normalised activity in the healthy group. We demonstrated that pulmonary blood vessel density and degree of emphysema were strongly correlated with this activity signal and identified as confounding factors, highlighting the need to address differences in target-organ characteristics in COPD. Experimental methods to adjust for these factors were developed for organ-specific signal quantification.

Conclusions: we report novel analysis techniques for molecular imaging of the human lung, presenting a platform which provides new insights into complex inflammatory disease and future precision medicine approaches.
2312-0541
Welham, Benjamin
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Bennett, Michael
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Ostridge, Kristoffer
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Guy, Matt
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Zvavamwe, Clint
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Chilcott, Anna
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Johns, Sandra
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Sundram, Francis
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Spalluto, Mirella Cosma
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Shaw, Emily
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Harden, Stephen
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Alzetani, Aiman
48518c15-14fa-4d9f-a472-d648e401444e
Lee, Paul
02620eab-ae7f-4a1c-bad1-8a50e7e48951
Lawson, Matthew John
5c14101b-e305-463d-97fd-d38b0000c3d6
Lackie, Peter
4afbbe1a-22a6-4ceb-8cad-f3696dc43a7a
Michopoulou, Sofia
f21ba2a3-f5d3-4998-801f-1ae72ff5d92c
Henley, Darren
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Kong, Chia Wei
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Fazleen, Aishath
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Cellura, Doriana
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McCrae, Christopher
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Platt, Adam
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Belvisi, Maria
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Staples, Karl J.
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Wilkinson, Tom
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Welham, Benjamin
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Bennett, Michael
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Ostridge, Kristoffer
d2271bae-b078-4390-8919-8f8c0e20542c
Guy, Matt
1a40b2ed-3aec-4fce-9954-396840471c28
Zvavamwe, Clint
a7537da6-3b05-47a7-8711-6ba3e5869ca9
Chilcott, Anna
c3449247-8cf0-44a2-9266-3ca128099be6
Johns, Sandra
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Sundram, Francis
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Spalluto, Mirella Cosma
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Shaw, Emily
adaae8b0-7d3b-4840-81aa-803cc86adde7
Harden, Stephen
f53e511e-df8b-451f-aa1e-e8e80e1a4e46
Alzetani, Aiman
48518c15-14fa-4d9f-a472-d648e401444e
Lee, Paul
02620eab-ae7f-4a1c-bad1-8a50e7e48951
Lawson, Matthew John
5c14101b-e305-463d-97fd-d38b0000c3d6
Lackie, Peter
4afbbe1a-22a6-4ceb-8cad-f3696dc43a7a
Michopoulou, Sofia
f21ba2a3-f5d3-4998-801f-1ae72ff5d92c
Henley, Darren
b2670616-2509-4419-918c-ca2c1e0f700b
Kong, Chia Wei
c187ab73-57ea-43c8-8482-a7279432c90a
Fazleen, Aishath
d96dba0e-f819-42cf-880f-ab927665b838
Cellura, Doriana
5edb82b2-f50c-4c76-bd10-8bf687a91b4d
McCrae, Christopher
905349d4-6151-412b-b146-7f1481d8472b
Platt, Adam
1cf7f1f0-5b57-407d-b6f1-51b5bebc204d
Belvisi, Maria
5db9e025-50e5-4433-84ae-e19a57402a1e
Staples, Karl J.
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Wilkinson, Tom
8c55ebbb-e547-445c-95a1-c8bed02dd652

Welham, Benjamin, Bennett, Michael, Ostridge, Kristoffer, Guy, Matt, Zvavamwe, Clint, Chilcott, Anna, Johns, Sandra, Sundram, Francis, Spalluto, Mirella Cosma, Shaw, Emily, Harden, Stephen, Alzetani, Aiman, Lee, Paul, Lawson, Matthew John, Lackie, Peter, Michopoulou, Sofia, Henley, Darren, Kong, Chia Wei, Fazleen, Aishath, Cellura, Doriana, McCrae, Christopher, Platt, Adam, Belvisi, Maria, Staples, Karl J. and Wilkinson, Tom (2025) A novel SPECT-CT imaging platform for quantifying in vivo lung cytokine signals in COPD. ERJ Open Research. (doi:10.1183/23120541.01246-2024).

Record type: Article

Abstract

Introduction: disease-modifying treatments such as monoclonal antibodies can be highly effective in chronic inflammatory diseases such as COPD, but often fail in clinical trials due to heterogeneity of inflammation and imperfect tools to stratify patients to select optimal therapeutic approaches. Molecular imaging provides the potential to transform precision medicine in this field.

Methods: we developed and tested a novel molecular imaging platform using therapeutic monoclonal antibodies labelled with SPECT-CT detectable markers to quantify in vivo TNF involved in chronic lung inflammation in humans. We undertook a proof-of-concept clinical study involving participants with COPD and healthy controls. Participants underwent SPECT-CT imaging at 6- and 24-hours following injection of 99m-Tc-anti-TNF. Segmentation of lung regions and 99m-Tc-anti-TNF activity quantification was undertaken using novel semi-automated and AI-driven approaches.

Results: a significant increase in normalised activity, representing increased TNF inflammatory activity, was seen between the two time-points in the COPD group (64.88% +/- [SD] 31.04, p=.029) and not in healthy controls (35.38% +/- 34.33, =.110). However, analysis at a single time-point revealed higher normalised activity in the healthy group. We demonstrated that pulmonary blood vessel density and degree of emphysema were strongly correlated with this activity signal and identified as confounding factors, highlighting the need to address differences in target-organ characteristics in COPD. Experimental methods to adjust for these factors were developed for organ-specific signal quantification.

Conclusions: we report novel analysis techniques for molecular imaging of the human lung, presenting a platform which provides new insights into complex inflammatory disease and future precision medicine approaches.

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Accepted/In Press date: 11 April 2025
e-pub ahead of print date: 24 July 2025

Identifiers

Local EPrints ID: 503291
URI: http://eprints.soton.ac.uk/id/eprint/503291
ISSN: 2312-0541
PURE UUID: 3a3f2f2d-ea6d-449f-a0fe-de4e9c79eb1c
ORCID for Matt Guy: ORCID iD orcid.org/0000-0002-6818-2010
ORCID for Mirella Cosma Spalluto: ORCID iD orcid.org/0000-0001-7273-0844
ORCID for Paul Lee: ORCID iD orcid.org/0000-0002-5729-6450
ORCID for Matthew John Lawson: ORCID iD orcid.org/0000-0003-0115-1698
ORCID for Peter Lackie: ORCID iD orcid.org/0000-0001-7138-3764
ORCID for Chia Wei Kong: ORCID iD orcid.org/0000-0002-8260-6967
ORCID for Karl J. Staples: ORCID iD orcid.org/0000-0003-3844-6457

Catalogue record

Date deposited: 28 Jul 2025 16:46
Last modified: 22 Aug 2025 02:37

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Contributors

Author: Benjamin Welham
Author: Michael Bennett
Author: Kristoffer Ostridge
Author: Matt Guy ORCID iD
Author: Clint Zvavamwe
Author: Anna Chilcott
Author: Sandra Johns
Author: Francis Sundram
Author: Mirella Cosma Spalluto ORCID iD
Author: Emily Shaw
Author: Stephen Harden
Author: Aiman Alzetani
Author: Paul Lee ORCID iD
Author: Matthew John Lawson ORCID iD
Author: Peter Lackie ORCID iD
Author: Sofia Michopoulou
Author: Darren Henley
Author: Chia Wei Kong ORCID iD
Author: Aishath Fazleen
Author: Doriana Cellura
Author: Christopher McCrae
Author: Adam Platt
Author: Maria Belvisi
Author: Karl J. Staples ORCID iD
Author: Tom Wilkinson

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